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W108

WAY-100635 maleate salt

Name: WAY-100635 maleate salt
Brand: SIGMA

5-HT1A serotonin receptor antagonist, powder

Synonym(s):

N-[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]-N-2-pyridinylcyclohexanecarboxamide maleate salt

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About This Item

Empirical Formula (Hill Notation):

C₂₅H₃₄N₄O₂ · C₄H₄O₄

CAS Number:

634908-75-1

Molecular Weight:

538.64

UNSPSC Code:

12352200

PubChem Substance ID:

24278113

NACRES:

NA.77

MDL number:

MFCD01321056

Form:

powder

Quality level:

100

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Properties

Product Name

WAY-100635 maleate salt, powder

form

powder

Quality Level

100

color

white

solubility

H₂O: 25 mg/mL

SMILES string

[H]\C(=C(/[H])C(O)=O)C(O)=O.COc1ccccc1N2CCN(CC2)CCN(C(=O)C3CCCCC3)c4ccccn4

InChI

1S/C25H34N4O2.C4H4O4/c1-31-23-12-6-5-11-22(23)28-18-15-27(16-19-28)17-20-29(24-13-7-8-14-26-24)25(30)21-9-3-2-4-10-21;5-3(6)1-2-4(7)8/h5-8,11-14,21H,2-4,9-10,15-20H2,1H3;1-2H,(H,5,6)(H,7,8)/b;2-1-

InChI key

XIGAHNVCEFUYOV-BTJKTKAUSA-N

Gene Information

human ... HTR1A(3350)

Description

Application

WAY-100635 maleate salt has been used as a 5-HT1A serotonin receptor antagonist:

to study whether the behavior of the cleaner wrasse is regulated by serotonin activity
to block activity of 3,4 methylenedioxymethamphetamine (MDMA) used to induce oxytocin release in male Wistar rats to increase their social behavior
to study the role of serotonin during metamorphosis of the ascidian Phallusia mammillata larvae

Biochem/physiol Actions

WAY-100635 maleate salt is a highly selective 5-HT1A serotonin receptor antagonist. It has an ability to inhibit brexpiprazole, an antipsychotic drug that regulates serotonin-dopamine activity.

Storage Class

11 - Combustible Solids

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

ppe

Eyeshields, Gloves, type N95 (US)

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